SCHEMBL3267285

SCHEMBL3267285

O[C@H](CNC1CC1)c1ccc(CN(Cc2nc3ccccc3[nH]2)C2CCCc3cccnc32)cc1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.72
CHRM2 P08172 1/20 0.61
CYP2D6 P10635 1/20 0.61
DRD2 P14416 1/20 0.61
OPRM1 P35372 1/20 0.61
KCNH2 Q12809 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3265558 0.89 CXCR4 (0.69) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL13909512 0.88 CXCR4 (0.91) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4791654 0.87 CXCR4 (0.63) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2506547 0.85 CXCR4 (0.83) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4932646 0.85 CXCR4 (0.85) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL3374214 0.85 CXCR4 (0.74) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2509563 0.85 CXCR4 (0.79) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4069355 0.84 CXCR4 (0.78) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2504776 0.84 CXCR4 (0.86) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2510467 0.84 CXCR4 (0.77) CXCR4CHRM2CYP2D6DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025416-A1 CXCR4 ANTAGONISTS FOR KIDNEY INJURY GENZYME CORPORATION (US) 2010-03-04 WO disclosed