SCHEMBL326738

SCHEMBL326738

COc1ccc(-c2nnc(C(=O)N3C[CH]C3)o2)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 17/20 0.58
KCNH2 Q12809 15/20 0.58
HRH3 Q9Y5N1 1/20 0.52
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL175935 0.84 MCHR1 (0.65) MCHR1KCNH2HRH3
SCHEMBL163159 0.79 MCHR1 (0.62) MCHR1KCNH2HRH3
SCHEMBL8840247 0.78 PTPN1 (0.68) NPC1RAB9AKMT2A
SCHEMBL17328846 0.78 MCHR1 (0.60) MCHR1KCNH2HRH3
SCHEMBL11222701 0.77 NPC1 (0.58) NPC1RAB9AKMT2A
SCHEMBL30968135 0.77 NPC1 (0.61) NPC1RAB9AKMT2A
SCHEMBL163155 0.77 MCHR1 (0.70) MCHR1KCNH2HRH3
SCHEMBL322320 0.74 MCHR1 (1.00) MCHR1KCNH2HRH3
SCHEMBL13004548 0.74 NPC1 (0.85) NPC1RAB9AKMT2A
SCHEMBL30968155 0.73 SMPD1 (0.61) NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590969-A2 THERAPEUTIC AGENTS 976 AstraZeneca AB (SE) 2013-05-15 EP disclosed
WO-2012004588-A2 THERAPEUTIC AGENTS 976 ASTRAZENECA AB (SE) 2012-01-12 WO disclosed