SCHEMBL3269409

SCHEMBL3269409

Cc1ccc(Cn2cnc3c(-c4ccco4)nc(N(C)C)nc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.60
ADORA1 P30542 13/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14429599 0.91 ADORA2A (0.61) ADORA2AADORA1
SCHEMBL3269836 0.90 ADORA2A (0.58) ADORA2AADORA1
SCHEMBL5467614 0.89 ADORA2A (0.75) ADORA2AADORA1
SCHEMBL3267585 0.86 ADORA2A (0.66) ADORA2AADORA1
SCHEMBL14429605 0.86 ADORA2A (0.63) ADORA2AADORA1
SCHEMBL3267851 0.85 ADORA2A (0.82) ADORA2AADORA1
SCHEMBL3268042 0.82 ADORA2A (0.59) ADORA2AADORA1
SCHEMBL3273511 0.82 ADORA2A (0.59) ADORA2AADORA1
SCHEMBL5461300 0.81 ADORA2A (0.56) ADORA2AADORA1
SCHEMBL14429601 0.78 ADORA2A (0.65) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-B1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2010-06-16 EP disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed