SCHEMBL3274138

SCHEMBL3274138

CS(=O)(=O)Nc1cccc(Cn2cnc3c(-c4ccco4)nc(N)nc32)c1

nearest known ligand 0.73

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.73
ADORA1 P30542 12/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3269182 0.91 ADORA2A (0.79) ADORA2AADORA1
SCHEMBL3268297 0.87 ADORA2A (0.72) ADORA2AADORA1
SCHEMBL3269034 0.86 ADORA2A (0.66) ADORA2AADORA1
SCHEMBL3269171 0.84 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL3268186 0.84 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL3268141 0.83 ADORA2A (0.69) ADORA2AADORA1
SCHEMBL3270162 0.83 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL3272671 0.82 ADORA2A (0.81) ADORA2AADORA1
SCHEMBL3268539 0.82 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL3274034 0.82 ADORA2A (0.81) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-B1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2010-06-16 EP disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed