SCHEMBL3274418

SCHEMBL3274418

Nc1nc(-c2ccco2)c2ncn(CC(=O)Nc3ccc(F)c(F)c3)c2n1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.58
ADORA1 P30542 12/20 0.58
ADORA3 P0DMS8 1/20 0.50
ADORA2B P29275 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3269823 0.88 ADORA2A (0.67) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3273089 0.88 ADORA2A (0.58) ADORA2AADORA1
SCHEMBL3269889 0.88 ADORA2A (0.65) ADORA2AADORA1
SCHEMBL3275259 0.87 ADORA2A (0.70) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3270073 0.85 ADORA2A (0.60) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3269070 0.83 ADORA2A (0.67) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3269210 0.83 ADORA2A (0.57) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3269452 0.83 ADORA2A (0.63) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3269023 0.81 ADORA2A (0.59) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3268791 0.81 ADORA2A (0.58) ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-B1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2010-06-16 EP disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed
US-7452894-B2 Purine derivatives as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2008-11-18 US disclosed