SCHEMBL3312482

SCHEMBL3312482

C=C(C)O[C@H](C(=O)O)c1c(C)cc2c(ccc(=O)n2Cc2ccccc2)c1-c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MDM2 Q00987 3/20 0.37
PTGES2 Q9H7Z7 4/20 0.37
PTGES O14684 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPK8 P45983 2/20 0.36
PLA2G10 O15496 1/20 0.36
MDM4 O15151 2/20 0.36
PSD A5PKW4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3311066 0.92 KDM4E (0.37) PTGDR2MEN1KMT2AMDM2PTGES2
SCHEMBL3297264 0.87 CYP3A4 (0.42) PTGDR2MEN1KMT2AMDM2PTGES2
SCHEMBL3312494 0.85 CYP3A4 (0.32) PTGDR2KDM4E
SCHEMBL15182599 0.84 PTGES2 (0.41) PTGDR2MEN1KMT2AMDM2PTGES2
SCHEMBL15186207 0.79 CYP3A4 (0.42) PTGES2PTGESKDM4E
SCHEMBL15093467 0.79 PPARG (0.43)
SCHEMBL15102812 0.79 PPARG (0.43)
SCHEMBL15102803 0.79 MAPK8 (0.39) PTGDR2PTGES2PTGESMAPK8PSD
SCHEMBL15093592 0.79 MAPK8 (0.39) PTGDR2PTGES2PTGESMAPK8PSD
SCHEMBL252857 0.78 PTGES2 (0.39) PTGDR2MEN1KMT2AMDM2PTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed