SCHEMBL3344824

SCHEMBL3344824

N#Cc1cccc(-c2nc(N)c3cc(CC(O)N4CCOCC4)sc3n2)c1

nearest known ligand 0.73

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.73
ADORA1 P30542 16/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301521 0.84 ADORA1 (1.00) ADORA2AADORA1
SCHEMBL3306497 0.83 ADORA2A (0.82) ADORA2AADORA1
SCHEMBL3350962 0.82 ADORA2A (0.74) ADORA2AADORA1
SCHEMBL13389826 0.81 ADORA2A (0.71) ADORA2AADORA1
SCHEMBL3304444 0.81 ADORA2A (0.71) ADORA2AADORA1
SCHEMBL2305928 0.78 ADORA1 (1.00) ADORA2AADORA1
SCHEMBL3300813 0.78 ADORA2A (0.67) ADORA2AADORA1
SCHEMBL3295339 0.78 ADORA2A (0.72) ADORA2AADORA1
SCHEMBL2304290 0.78 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL2301454 0.77 ADORA1 (1.00) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045016-A1 HETEROCYCLYL AND CYCLOALKYL SUBSTITUTED THIENO [2,3-D] PYRIMIDINE AND THEIR USE AS ADENOSINE A2A RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-04-22 WO disclosed