SCHEMBL3346791

SCHEMBL3346791

COc1cc(N(C)C(=O)C2CCNCC2)ccc1Nc1ncc(Cl)c(-c2cnc3c(F)cccn23)n1

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 20/20 0.63
KCNH2 Q12809 9/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3318526 0.87 IGF1R (0.64) IGF1RKCNH2
SCHEMBL3313499 0.84 IGF1R (0.76) IGF1RKCNH2
SCHEMBL3311216 0.83 IGF1R (0.67) IGF1RKCNH2
SCHEMBL3315964 0.83 IGF1R (0.68) IGF1RKCNH2
SCHEMBL3311801 0.83 IGF1R (0.66) IGF1RKCNH2
SCHEMBL3314225 0.82 IGF1R (0.64) IGF1RKCNH2
SCHEMBL3309415 0.81 IGF1R (0.64) IGF1RKCNH2
SCHEMBL3314782 0.81 IGF1R (0.62) IGF1RKCNH2
SCHEMBL3316240 0.81 IGF1R (0.61) IGF1RKCNH2
SCHEMBL3317767 0.80 IGF1R (0.80) IGF1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010049731-A1 PYRAZOLO- AND IMIDAZOPYRIDINYLPYRIMIDINEAMINES AS IGF-1R TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-05-06 WO disclosed