SCHEMBL3353023

SCHEMBL3353023

COc1cccc([C@H](C)N)n1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.54
CD274 Q9NZQ7 5/20 0.40
PDCD1LG2 Q9BQ51 3/20 0.40
HRH1 P35367 1/20 0.39
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 1/20 0.38
PDCD1 Q15116 2/20 0.38
IDH1 O75874 1/20 0.37
BTK Q06187 1/20 0.37
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30824556 1.00 TAAR1 (0.54) TAAR1CD274PDCD1LG2HRH1CYP3A4
SCHEMBL2936969 1.00 TAAR1 (0.54) TAAR1CD274PDCD1LG2HRH1CYP3A4
SCHEMBL29793607 1.00 TAAR1 (0.54) TAAR1CD274PDCD1LG2HRH1CYP3A4
SCHEMBL18793289 1.00 TAAR1 (0.54) TAAR1CD274PDCD1LG2HRH1CYP3A4
Hydrochloric Acid SCHEMBL15994343 0.98 TAAR1 (0.52) TAAR1CD274PDCD1LG2HRH1CYP3A4
SCHEMBL179528 0.83 TAAR1 (0.42) TAAR1HRH1CYP3A4CYP2D6SLC6A2
SCHEMBL29337164 0.82 TAAR1 (0.43) TAAR1HRH1CYP3A4CYP2D6SLC6A2
SCHEMBL522063 0.80 CYP1A2 (0.38) TAAR1CD274PDCD1LG2CYP3A4CYP2D6
SCHEMBL38661915 0.80 CYP3A4 (0.44) TAAR1HRH1CYP3A4CYP2D6SLC6A2
SCHEMBL4196024 0.80 CYP3A4 (0.44) TAAR1HRH1CYP3A4CYP2D6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed