SCHEMBL3361841

SCHEMBL3361841

COc1cncc(-c2cc3c(c(Nc4ccc(N5C[C@@H](C)O[C@@H](C)C5)nc4)n2)C(=O)[N]C=C3)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.39
ZAP70 P43403 2/20 0.38
BTK Q06187 1/20 0.36
KCNH2 Q12809 1/20 0.36
SYK P43405 4/20 0.35
PIK3CA P42336 2/20 0.33
GAK O14976 1/20 0.32
SMO Q99835 2/20 0.31
PGR P06401 1/20 0.31
GPR183 P32249 1/20 0.31
DYRK1A Q13627 2/20 0.31
CLK2 P49760 1/20 0.31
CLK3 P49761 1/20 0.31
WNT1 P04628 1/20 0.31
TYK2 P29597 1/20 0.30
PIK3CD O00329 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361973 0.80 ZAP70 (0.47) LRRK2ZAP70SYKTYK2
SCHEMBL1049202 0.79 ZAP70 (0.61) LRRK2ZAP70BTKKCNH2SYK
SCHEMBL3362641 0.79 PIK3CA (0.38) BTKKCNH2SYKPIK3CASMO
SCHEMBL3357809 0.77 SYK (0.44) ZAP70BTKKCNH2SYKPIK3CA
SCHEMBL3359856 0.76 ZAP70 (0.40) ZAP70SYKPIK3CAPIK3CDPIK3CB
SCHEMBL3360026 0.76 SYK (0.46) LRRK2ZAP70BTKKCNH2SYK
SCHEMBL3358811 0.76 SYK (0.46) LRRK2ZAP70BTKKCNH2SYK
SCHEMBL3362887 0.75 ZAP70 (0.46) ZAP70BTKSYK
SCHEMBL3361678 0.75 ZAP70 (0.42) ZAP70SYK
SCHEMBL3359641 0.75 ZAP70 (0.41) ZAP70SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238137-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2010-10-13 EP claimed
WO-2009097287-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2009-08-06 WO claimed