SCHEMBL3366966

SCHEMBL3366966

COc1ccc(CC(=O)NCc2nc3cc(C=CC(=O)NO)ccc3n2C)cc1

nearest known ligand 0.80

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 19/20 0.80
HDAC8 Q9BY41 9/20 0.58
HDAC2 Q92769 2/20 0.55
HDAC11 Q96DB2 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC3 O15379 1/20 0.52
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366963 1.00 HDAC1 (0.80) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL13227295 0.93 HDAC1 (0.69) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL3368738 0.89 HDAC1 (1.00) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL3368735 0.89 HDAC1 (1.00) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL3372393 0.89 HDAC1 (1.00) HDAC1HDAC8
SCHEMBL3372397 0.89 HDAC1 (1.00) HDAC1HDAC8
SCHEMBL3369172 0.88 HDAC1 (1.00) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL3369167 0.88 HDAC1 (1.00) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL16788426 0.87 HDAC1 (0.75) HDAC1HDAC8HDAC2HDAC11HDAC6
SCHEMBL13226894 0.83 HDAC1 (0.82) HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673349-B1 BENZIMIDAZOLE DERIVATIVES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S BIO PTE LTD (SG) 2010-06-30 EP claimed