SCHEMBL3368078

SCHEMBL3368078

CCCc1ccc(C(=O)N2CCCC2c2nnc(-c3cccc(OC)c3)o2)cc1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 9/20 0.61
HCRTR2 O43614 9/20 0.61
SCD5 Q86SK9 1/20 0.47
GRM5 P41594 2/20 0.46
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.44
ROCK2 O75116 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3367057 0.88 HCRTR1 (0.65) HCRTR1HCRTR2SCD5GRM5NPC1
SCHEMBL3366784 0.88 HCRTR1 (0.65) HCRTR1HCRTR2SCD5GRM5ROCK2
SCHEMBL3367000 0.86 HCRTR1 (0.54) HCRTR1HCRTR2GRM5TP53MAPT
SCHEMBL3368112 0.85 HCRTR1 (0.61) HCRTR1HCRTR2SCD5GRM5
SCHEMBL3364799 0.83 HCRTR1 (0.64) HCRTR1HCRTR2SCD5GRM5NPC1
SCHEMBL3368411 0.83 HCRTR1 (0.61) HCRTR1HCRTR2SCD5GRM5NPC1
SCHEMBL3366762 0.83 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL3369692 0.83 HCRTR1 (0.59) HCRTR1HCRTR2GRM5NPC1RAB9A
SCHEMBL3368150 0.83 HCRTR1 (0.67) HCRTR1HCRTR2SCD5GRM5MAPT
SCHEMBL3366720 0.82 HCRTR1 (0.65) HCRTR1HCRTR2SCD5GRM5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-B1 2-PYRROLIDIN-2-YL- [1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS GRUENENTHAL GMBH (DE) 2010-10-13 EP disclosed