SCHEMBL3368889

SCHEMBL3368889

O=C(O)[C@H]1CC(=O)N(c2ccc(OCc3ccc(F)cc3)cc2)C1

nearest known ligand 0.81

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.81
RAB9A P51151 6/20 0.81
POLB P06746 3/20 0.81
HPGD P15428 2/20 0.66
KMT2A Q03164 3/20 0.64
GLA P06280 1/20 0.64
S1PR5 Q9H228 1/20 0.62
FFAR1 O14842 1/20 0.61
ALDH1A1 P00352 3/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56
TSHR P16473 1/20 0.54
HTT P42858 1/20 0.54
MEN1 O00255 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3365549 1.00 NPC1 (0.81) NPC1RAB9APOLBHPGDKMT2A
SCHEMBL3365543 1.00 NPC1 (0.81) NPC1RAB9APOLBHPGDKMT2A
SCHEMBL3369373 0.89 GLA (0.75) NPC1RAB9APOLBHPGDKMT2A
SCHEMBL3363933 0.89 GLA (0.75) NPC1RAB9APOLBHPGDKMT2A
SCHEMBL3363939 0.89 GLA (0.75) NPC1RAB9APOLBHPGDKMT2A
SCHEMBL3365348 0.88 NPC1 (0.77) NPC1RAB9APOLBKMT2AALDH1A1
SCHEMBL3365355 0.88 NPC1 (0.77) NPC1RAB9APOLBKMT2AALDH1A1
SCHEMBL3366005 0.88 NPC1 (0.77) NPC1RAB9APOLBKMT2AALDH1A1
SCHEMBL3363108 0.87 NPC1 (0.78) NPC1RAB9APOLBKMT2AALDH1A1
SCHEMBL3363165 0.87 NPC1 (0.78) NPC1RAB9APOLBKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542970-B1 PYRROLIDONE DERIVATIVES AS MAOB INHIBITORS HOFFMANN LA ROCHE (CH) 2010-06-30 EP disclosed
US-7151111-B2 4-pyrrolidino-phenyl-benzyl ether derivatives HOFFMANN-LA ROCHE INC. (US) 2006-12-19 US disclosed
EP-1542970-A1 PYRROLIDONE DERIVATIVES AS MAOB INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2005-06-22 EP disclosed
US-20040116707-A1 4-Pyrrolidino-phenyl-benzyl ether derivatives HOFFMANN-LA ROCHE INC. 2004-06-17 US disclosed
WO-2004026825-A1 PYRROLIDONE DERIVATIVES AS MAOB INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2004-04-01 WO disclosed