SCHEMBL3370704

SCHEMBL3370704

COc1cccc(-c2nnc(C3CCCN3C(=O)c3nn(-c4ccccc4)nc3C)o2)c1

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.63
HCRTR2 O43614 19/20 0.63
SCD5 Q86SK9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366040 0.85 HCRTR1 (0.56) HCRTR1HCRTR2
SCHEMBL3368150 0.82 HCRTR1 (0.67) HCRTR1HCRTR2SCD5
SCHEMBL3368066 0.80 HCRTR1 (0.71) HCRTR1HCRTR2SCD5
SCHEMBL3366784 0.79 HCRTR1 (0.65) HCRTR1HCRTR2SCD5
SCHEMBL3367057 0.79 HCRTR1 (0.65) HCRTR1HCRTR2SCD5
SCHEMBL3366720 0.79 HCRTR1 (0.65) HCRTR1HCRTR2SCD5
SCHEMBL3366800 0.79 HCRTR1 (0.65) HCRTR1HCRTR2
SCHEMBL3366717 0.78 HCRTR1 (0.68) HCRTR1HCRTR2SCD5
SCHEMBL3364799 0.78 HCRTR1 (0.64) HCRTR1HCRTR2SCD5
SCHEMBL17063859 0.77 HCRTR1 (1.00) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-B1 2-PYRROLIDIN-2-YL- [1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS GRUENENTHAL GMBH (DE) 2010-10-13 EP disclosed