SCHEMBL3375347

SCHEMBL3375347

O=C1CNc2nccc(OCc3ccccc3)c2N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.44
CREBBP Q92793 2/20 0.44
HTT P42858 2/20 0.43
TNKS2 Q9H2K2 1/20 0.41
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
LTA4H P09960 1/20 0.39
MAPK14 Q16539 1/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TTR P02766 1/20 0.39
BLM P54132 1/20 0.39
PLA2G1B P04054 1/20 0.39
POLB P06746 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
LMNA P02545 1/20 0.39
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7211895 0.70 BRD4 (0.53) BRD4CREBBPHTTCYP19A1CYP11B1
SCHEMBL2933275 0.69 BRAF (0.41) MAPK14BRAF
SCHEMBL16536586 0.69 PDE4A (0.53) BRD4CREBBPCYP19A1CYP11B1CYP11B2
SCHEMBL16537757 0.69 PDE4A (0.53) BRD4CREBBPCYP19A1CYP11B1CYP11B2
SCHEMBL25366826 0.68 HTT (0.42) BRD4CREBBPHTTPOLBLMNA
SCHEMBL16563587 0.68 PDE3A (0.36) BRD4CREBBPALDH1A1POLBLMNA
SCHEMBL4894335 0.68 BRD4 (0.50) BRD4CREBBPHTTMEN1ALDH1A1
SCHEMBL6074738 0.67 BRD4 (0.46) BRD4CREBBPCYP19A1CYP11B1CYP11B2
SCHEMBL22368749 0.67 BRD4 (0.61) BRD4CREBBPHTTTNKS2CYP19A1
SCHEMBL5546557 0.67 BRD4 (0.46) BRD4CREBBPHTTCYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed