SCHEMBL337699

SCHEMBL337699

COC[C@H]1C[C@H](CC(=O)NC2CCC(CCN3CCC(C(=O)c4ccc(F)cc4)CC3)CC2)C1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 7/20 0.49
HTR2A P28223 6/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
LMNA P02545 2/20 0.48
HTT P42858 1/20 0.48
HTR2C P28335 1/20 0.47
HTR7 P34969 1/20 0.47
HTR6 P50406 1/20 0.47
ALDH1A1 P00352 1/20 0.47
DRD4 P21917 2/20 0.46
HTR1A P08908 1/20 0.46
DRD2 P14416 1/20 0.46
HTR2B P41595 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1923273 1.00 DRD3 (0.49) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL10086739 1.00 DRD3 (0.49) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL1923651 1.00 DRD3 (0.49) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL1923274 1.00 DRD3 (0.49) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL337028 1.00 DRD3 (0.49) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL1923275 1.00 DRD3 (0.49) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL337609 0.97 HTR2A (0.48) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL337607 0.97 HTR2A (0.48) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL337608 0.97 HTR2A (0.48) DRD3HTR2ASMN1; SMN2LMNAHTT
SCHEMBL337024 0.95 HTR2A (0.53) DRD3HTR2ASMN1; SMN2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097637-B2 Benzoyl-piperidine derivatives as dual modulators of the 5-HT2A and D3 receptors HOFFMANN-LA ROCHE INC. (US) 2012-01-17 US claimed
EP-2185513-B1 BENZOYL-PIPERIDINE DERIVATIVES AS DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2011-06-08 EP claimed
US-8097637-B2 Benzoyl-piperidine derivatives as dual modulators of the 5-HT2A and D3 receptors HOFFMANN-LA ROCHE INC. (US) 2012-01-17 US disclosed
EP-2185513-B1 BENZOYL-PIPERIDINE DERIVATIVES AS DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2011-06-08 EP disclosed