SCHEMBL3377095

SCHEMBL3377095

O[C@@]1(C#Cc2cccc(Cl)c2)C[CH]CCC1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.44
PTGES O14684 2/20 0.38
KCNH2 Q12809 1/20 0.38
MAP3K14 Q99558 1/20 0.35
NPC1 O15118 4/20 0.34
RAB9A P51151 4/20 0.34
POLB P06746 1/20 0.34
NR2F2 P24468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052069 0.76 GRM5 (0.46) GRM5PTGESKCNH2MAP3K14NPC1
SCHEMBL5123963 0.76 GRM5 (0.43) GRM5PTGESKCNH2MAP3K14
SCHEMBL5115607 0.75 GRM5 (0.46) GRM5PTGESKCNH2MAP3K14
SCHEMBL3276812 0.74 GRM5 (0.49) GRM5PTGESKCNH2MAP3K14
SCHEMBL1899368 0.74 GRM5 (0.49) GRM5PTGESKCNH2MAP3K14
SCHEMBL3840451 0.74 GRM5 (0.48) GRM5KCNH2NPC1RAB9APOLB
SCHEMBL4046766 0.73 GRM5 (0.41) GRM5PTGESKCNH2MAP3K14NPC1
SCHEMBL3838272 0.72 GRM5 (0.50) GRM5PTGESKCNH2MAP3K14
SCHEMBL3839812 0.72 GRM5 (0.50) GRM5PTGESKCNH2MAP3K14
SCHEMBL5128660 0.72 GRM5 (0.44) GRM5PTGESKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877365-B1 ACETYLENE DERIVATIVES NOVARTIS AG (CH) 2010-11-10 EP claimed