SCHEMBL3377792

SCHEMBL3377792

COc1cccc2c([C@@H](O)[C@H](O)C3CCC(NCc4ccc5c(n4)NC(=O)CO5)CC3)ccnc12

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.50
KCNQ1 P51787 1/20 0.44
CACNA1C Q13936 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5253483 0.86 KCNH2 (0.54) KCNH2KCNQ1CACNA1C
SCHEMBL3378200 0.85 KCNH2 (0.44) KCNH2
SCHEMBL16649510 0.84 KCNH2 (0.53) KCNH2KCNQ1CACNA1C
SCHEMBL3377361 0.84 KCNH2 (0.69) KCNH2KCNQ1CACNA1C
SCHEMBL3377367 0.84 KCNH2 (0.69) KCNH2KCNQ1CACNA1C
SCHEMBL3376441 0.82 KCNH2 (0.55) KCNH2KCNQ1CACNA1C
SCHEMBL3376444 0.82 KCNH2 (0.55) KCNH2KCNQ1CACNA1C
SCHEMBL3373011 0.82 KCNH2 (0.55) KCNH2KCNQ1CACNA1C
SCHEMBL3373008 0.82 KCNH2 (0.55) KCNH2KCNQ1CACNA1C
SCHEMBL3377415 0.75 KCNH2 (0.44) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987040-B1 ETHANOL OR 1,2-ETHANEDIOL CYCLOHEXYL ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-11-10 EP claimed