SCHEMBL3379845

SCHEMBL3379845

O=C(NCC1CCC1)Oc1cnc(Nc2ccc(C(F)(F)F)c(F)c2)nc1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 17/20 0.52
CYP2C19 P33261 6/20 0.52
CYP3A4 P08684 6/20 0.52
CYP2C9 P11712 6/20 0.52
CYP1A2 P05177 5/20 0.52
CYP2D6 P10635 4/20 0.52
PLK4 O00444 2/20 0.40
CHEK1 O14757 2/20 0.40
AURKA O14965 2/20 0.40
PRKD3 O94806 2/20 0.40
MAP4K4 O95819 2/20 0.40
PAK4 O96013 2/20 0.40
ABL1 P00519 2/20 0.40
NTRK1 P04629 2/20 0.40
INSR P06213 2/20 0.40
FES P07332 2/20 0.40
RET P07949 2/20 0.40
IGF1R P08069 2/20 0.40
MET P08581 2/20 0.40
FGFR1 P11362 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379074 0.92 CNR2 (0.57) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3380884 0.89 CNR2 (0.58) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3382843 0.87 CNR2 (0.58) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3380806 0.87 CNR2 (0.62) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3383217 0.87 CNR2 (0.59) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3378862 0.86 CNR2 (0.60) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3379885 0.86 CNR2 (0.58) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3382577 0.85 CNR2 (0.59) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3382325 0.85 CNR2 (0.62) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3378861 0.85 CNR2 (0.71) CNR2CYP2C19CYP3A4CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878725-B1 Pyrimidine derivatives and their use as CB2 modulators GLAXO GROUP LTD (GB) 2010-11-24 EP claimed