SCHEMBL3380729

SCHEMBL3380729

CN(C)Cc1ccc(-c2ccn3c(-c4ccc(CNC(=O)Nc5cccc(C(F)(F)F)c5)cc4)cnc3c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KDR P35968 19/20 0.57
FGFR3 P22607 17/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386228 0.93 KDR (0.55) KDRFGFR3
SCHEMBL3383984 0.90 KDR (0.68) KDRFGFR3
SCHEMBL3187562 0.88 KDR (0.56) KDRFGFR3
SCHEMBL3185744 0.87 KDR (0.57) KDRFGFR3
SCHEMBL3184677 0.87 FGFR3 (0.57) KDRFGFR3
SCHEMBL3382522 0.87 KDR (0.53) KDRFGFR3
SCHEMBL3380727 0.86 KDR (0.70) KDRFGFR3
SCHEMBL3187469 0.86 FGFR3 (0.59) KDRFGFR3
SCHEMBL3382054 0.86 KDR (0.55) KDRFGFR3
SCHEMBL3384511 0.86 KDR (0.55) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed