SCHEMBL3380867

SCHEMBL3380867

Cc1cc(Cn2c(C)c(C(=O)N[C@H](c3cccc(F)c3)C3CCC3)c3c([C@@H](c4cccc(F)c4C(N)=O)C4CCC4)ccc(F)c3c2=O)nn1C

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.36
TACR3 P29371 10/20 0.35
WDR5 P61964 3/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2310390 0.88 CYP2C9 (0.39) CYP2C9TACR3
SCHEMBL2356247 0.87 MAPT (0.31) GRIN1GRIN2B
SCHEMBL2306426 0.86 CYP2C9 (0.35) CYP2C9TACR3WDR5
SCHEMBL1366381 0.85 CYP2C9 (0.45) CYP2C9TACR3WDR5GRIN1GRIN2B
SCHEMBL3235809 0.85 CYP2C9 (0.39) CYP2C9TACR3
SCHEMBL2312871 0.84 CYP2C9 (0.39) CYP2C9TACR3WDR5
SCHEMBL2148919 0.84 CYP2C9 (0.39) CYP2C9TACR3WDR5
SCHEMBL2149069 0.82 CYP2C9 (0.36) CYP2C9TACR3
SCHEMBL3379662 0.82 CYP2C9 (0.36) CYP2C9TACR3
SCHEMBL2149246 0.81 CYP2C9 (0.35) CYP2C9TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045948-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-04-29 WO claimed