SCHEMBL3380913

SCHEMBL3380913

Cc1ccc(Nc2ncc(OC(=O)NCC3CCCCC3)c(C(F)(F)F)n2)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 18/20 0.54
CYP2C9 P11712 7/20 0.49
CYP3A4 P08684 6/20 0.49
CYP2C19 P33261 5/20 0.49
CYP1A2 P05177 5/20 0.48
CYP2D6 P10635 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379863 0.92 CNR2 (0.63) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3382328 0.92 CNR2 (0.54) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3383470 0.91 CNR2 (0.64) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3378175 0.91 CNR2 (0.62) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3379050 0.89 CNR2 (0.55) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3381103 0.88 CNR2 (0.63) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3381376 0.88 CNR2 (0.66) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3379227 0.88 CNR2 (0.52) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3381320 0.87 CNR2 (0.54) CNR2CYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL3383612 0.87 CNR2 (0.64) CNR2CYP2C9CYP3A4CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878725-B1 Pyrimidine derivatives and their use as CB2 modulators GLAXO GROUP LTD (GB) 2010-11-24 EP claimed