SCHEMBL3382983

SCHEMBL3382983

O=C(NCc1cccc(-c2cnc3cc(-c4ccncc4)ccn23)c1)Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.72

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.72
FGFR3 P22607 17/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383252 0.93 KDR (0.69) KDRFGFR3
SCHEMBL3383984 0.93 KDR (0.68) KDRFGFR3
SCHEMBL3380727 0.86 KDR (0.70) KDRFGFR3
SCHEMBL3383012 0.86 KDR (0.63) KDRFGFR3
SCHEMBL3190830 0.85 KDR (0.66) KDRFGFR3
SCHEMBL3197653 0.84 KDR (0.62) KDRFGFR3
SCHEMBL11908958 0.84 KDR (1.00) KDRFGFR3
SCHEMBL3383459 0.83 FGFR3 (0.61) KDRFGFR3
SCHEMBL3195980 0.82 RET (0.60) KDRFGFR3
SCHEMBL3384511 0.82 KDR (0.55) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed