SCHEMBL3384801

SCHEMBL3384801

COc1ccc(F)c(F)c1C(=O)c1sc(NC2CCN(C(=O)O)CC2)nc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 8/20 0.51
CDK4 P11802 7/20 0.51
CCND1 P24385 7/20 0.51
CDK5 Q00535 4/20 0.51
CDK1 P06493 4/20 0.51
CDK9 P50750 4/20 0.51
CDK6 Q00534 4/20 0.51
CDK11A Q9UQ88 4/20 0.51
DYRK1A Q13627 2/20 0.51
CLK1 P49759 2/20 0.51
CASK O14936 1/20 0.51
ROCK2 O75116 1/20 0.51
CDKL5 O76039 1/20 0.51
STK10 O94804 1/20 0.51
CDK14 O94921 1/20 0.51
ABL1 P00519 1/20 0.51
EGFR P00533 1/20 0.51
MAK P20794 1/20 0.51
CDK11B P21127 1/20 0.51
TTK P33981 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3389143 0.89 CDK2 (0.62) CDK2CDK4CCND1CDK5CDK1
SCHEMBL3386067 0.88 CDK2 (0.67) CDK2CDK4CCND1CDK5CDK1
SCHEMBL3385078 0.86 CDK5 (0.58) CDK2CDK4CCND1CDK5CDK1
SCHEMBL3386123 0.86 MEN1 (0.52) CDK2CDK5DYRK1ACLK1GSK3A
SCHEMBL3389148 0.85 CDK2 (0.49) CDK2CDK4CCND1CDK5CDK1
Formaldehyde SCHEMBL5005032 0.85 CDK5 (0.56) CDK2CDK4CCND1CDK5CDK1
SCHEMBL6197111 0.83 CDK5 (0.55) CDK2CDK4CCND1CDK5CDK1
Formaldehyde SCHEMBL3387471 0.82 CDK2 (0.60) CDK2CDK4CCND1CDK5CDK1
SCHEMBL3837802 0.81 CDK1 (0.58) CDK2CDK4CCND1CDK5CDK1
SCHEMBL3386135 0.79 CDK2 (0.51) CDK2CDK4CCND1CDK5CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771424-B1 NOVEL 2,4-DIAMINOTHIAZOL-5-ONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-15 EP claimed