SCHEMBL3387119

SCHEMBL3387119

CC(C)(C)C(CN)Nc1nc(Cl)c(C#N)cc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.47
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.32
PGK1 P00558 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
JAK2 O60674 2/20 0.31
JAK3 P52333 2/20 0.31
ACHE P22303 4/20 0.31
BCHE P06276 3/20 0.31
LIMK1 P53667 1/20 0.31
LIMK2 P53671 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP2D6 P10635 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
NOS2 P35228 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14910220 1.00 KHK (0.47) KHKALDH1A1PKMPGK1CYP1A2
SCHEMBL14928602 0.89 KHK (0.44) KHKALDH1A1PKMPGK1CYP1A2
SCHEMBL14677257 0.88 KHK (0.43) KHKALDH1A1PGK1CYP1A2CYP2C9
SCHEMBL14677256 0.88 KHK (0.43) KHKALDH1A1PGK1CYP1A2CYP2C9
SCHEMBL14685132 0.85 KHK (0.42) KHKALDH1A1PGK1CYP1A2CYP2C9
SCHEMBL14911090 0.84 KHK (0.48) KHKALDH1A1PKMPGK1CYP1A2
SCHEMBL14911089 0.84 KHK (0.48) KHKALDH1A1PKMPGK1CYP1A2
SCHEMBL14909860 0.83 KHK (0.50) KHKALDH1A1PKMPGK1CYP1A2
SCHEMBL14909858 0.83 KHK (0.50) KHKALDH1A1PKMPGK1CYP1A2
SCHEMBL19325112 0.82 KHK (0.39) KHKALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2589592-B1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM CORP (JP) 2018-08-22 EP disclosed
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-8772320-B2 2014-07-08 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed
WO-2012002577-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF 富士フイルム株式会社 (JP) 2012-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK KHK 2008/4885ALDH1A1 1638/4885PKM 3583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.