SCHEMBL3388616

SCHEMBL3388616

C[C@@H]1CN(Cc2ccc(F)cc2)CCN1C(=O)CC1CN(C(=O)O)c2cc(Cl)ccc2O1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 16/20 0.54
PTGDR2 Q9Y5Y4 2/20 0.51
FPR3 P25089 1/20 0.50
GPR65 Q8IYL9 1/20 0.50
GPR35 Q9HC97 1/20 0.50
ENPP2 Q13822 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3358218 0.89 CCR1 (0.51) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3358210 0.89 CCR1 (0.51) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3355002 0.82 CCR1 (0.54) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3355449 0.82 CCR1 (0.54) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3353758 0.78 CCR1 (0.53) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3353757 0.78 CCR1 (0.53) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3355615 0.76 CCR1 (0.49) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3355628 0.76 CCR1 (0.49) CCR1PTGDR2FPR3GPR65GPR35
Chlorobenzene SCHEMBL27693442 0.73 CCR1 (0.66) CCR1PTGDR2FPR3GPR65GPR35
SCHEMBL3354632 0.73 CCR1 (0.53) CCR1PTGDR2FPR3GPR65GPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068881-A1 NOVEL BENZODIOXANE AND BENZOXAZINE DERIVATIVES USEFUL AS CC CHEMOKINE RECEPTOR LIGANDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-06-17 WO disclosed