SCHEMBL3388925

SCHEMBL3388925

CC(C)N1CCN(C(=O)c2ccc3c(ccn3CC3CCCN(C(=O)O)C3)c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 11/20 0.45
CHRNA7 P36544 2/20 0.42
OXTR P30559 3/20 0.41
KDM4E B2RXH2 1/20 0.40
PADI4 Q9UM07 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387634 0.91 HRH3 (0.44) HRH3CHRNA7OXTRPADI4
SCHEMBL3944012 0.89 HRH3 (0.47) HRH3CHRNA7OXTR
SCHEMBL3948632 0.88 HRH3 (0.47) HRH3CHRNA7
SCHEMBL3387874 0.88 HRH3 (0.44) HRH3CHRNA7OXTR
SCHEMBL3390207 0.88 HRH3 (0.43) HRH3CHRNA7OXTR
SCHEMBL3390210 0.88 HRH3 (0.43) HRH3CHRNA7OXTR
SCHEMBL3390065 0.88 HRH3 (0.43) HRH3CHRNA7OXTR
SCHEMBL3388747 0.86 HRH3 (0.43) HRH3CHRNA7OXTR
SCHEMBL3388045 0.86 HRH3 (0.52) HRH3CHRNA7OXTR
SCHEMBL3390069 0.86 HRH3 (0.50) HRH3OXTRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029534-B1 1H-INDOL-5-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-22 EP disclosed