SCHEMBL3389138

SCHEMBL3389138

CCOC(=O)CC(CN)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
GAA P10253 2/20 0.40
MGAM O43451 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
ALDH1A1 P00352 7/20 0.38
TRPA1 O75762 1/20 0.38
ALOX15 P16050 3/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
HSD17B10 Q99714 2/20 0.35
CHRM1 P11229 1/20 0.35
ADORA1 P30542 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.32
CYP2D6 P10635 1/20 0.32
F2 P00734 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1262979 0.98 CYP1A2 (0.40) CYP1A2GAAMGAMSIMGAM2
SCHEMBL8668654 0.88 GAA (0.46) CYP1A2GAAMGAMSIMGAM2
Hydrochloric Acid SCHEMBL1260836 0.86 CYP1A2 (0.43) CYP1A2GAAMGAMSIMGAM2
SCHEMBL1129987 0.85 GAA (0.43) CYP1A2GAAMGAMSIMGAM2
SCHEMBL31252242 0.81 GAA (0.40) CYP1A2GAAMGAMSIMGAM2
SCHEMBL27383612 0.81 GAA (0.40) CYP1A2GAAMGAMSIMGAM2
SCHEMBL9419145 0.80 CA1 (0.42) CYP1A2GAAMGAMSIMGAM2
SCHEMBL28923720 0.79 GAA (0.38) CYP1A2GAAMGAMSIMGAM2
SCHEMBL28232656 0.79 GAA (0.38) CYP1A2GAAMGAMSIMGAM2
SCHEMBL5183401 0.77 GAA (0.43) CYP1A2GAAMGAMSIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863812-B1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD (KR) 2010-07-14 EP disclosed
EP-1863812-A4 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD (KR) 2009-06-24 EP disclosed
EP-1863812-A1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG Life Sciences Ltd. (KR) 2007-12-12 EP disclosed
WO-2006104356-A1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES, LTD. (KR) 2006-10-05 WO disclosed