SCHEMBL3392985

SCHEMBL3392985

NC(=O)N(c1ccc(F)cc1)c1ccc(-c2cccc3[nH]nc(N)c23)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.72
ABL1 P00519 7/20 0.72
LCK P06239 5/20 0.72
CSF1R P07333 5/20 0.72
FLT1 P17948 4/20 0.72
FGFR1 P11362 3/20 0.72
PRKACA P17612 3/20 0.72
ROCK1 Q13464 3/20 0.72
NTRK1 P04629 2/20 0.72
MET P08581 2/20 0.72
GSK3A P49840 2/20 0.72
GSK3B P49841 2/20 0.72
RPS6KA3 P51812 2/20 0.72
CDK5 Q00535 2/20 0.72
DYRK1A Q13627 2/20 0.72
DAPK3 O43293 1/20 0.72
PRKD3 O94806 1/20 0.72
MAP4K4 O95819 1/20 0.72
PAK4 O96013 1/20 0.72
RET P07949 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3363647 0.91 KDR (0.68) KDRABL1LCKCSF1RFLT1
SCHEMBL27657352 0.91 KDR (0.66) KDRABL1LCKCSF1RFLT1
SCHEMBL4737713 0.87 KDR (0.77) KDRABL1LCKCSF1RFLT1
SCHEMBL27825044 0.86 KDR (0.76) KDRABL1LCKCSF1RFLT1
SCHEMBL4739859 0.85 KDR (0.63) KDRABL1LCKCSF1RFLT1
SCHEMBL27657344 0.85 KDR (0.69) KDRABL1LCKCSF1RFLT1
SCHEMBL27636418 0.85 KDR (0.66) KDRABL1LCKCSF1RFLT1
SCHEMBL27636364 0.85 KDR (0.68) KDRABL1LCKCSF1RFLT1
SCHEMBL27636372 0.85 KDR (0.65) KDRABL1LCKCSF1RFLT1
SCHEMBL4740070 0.84 KDR (0.62) KDRABL1LCKCSF1RFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN claimed
EP-1638941-B1 INDAZOLE, BENZISOXAZOLE, AND BENZISOTHIAZOLE KINASE INHIBITORS ABBOTT LAB (US) 2010-06-02 EP claimed
WO-2008080110-A1 METHODS FOR TREATING MACULAR EDEMA AND PATHOLOGIC OCULAR ANGIOGENESIS USING A NEUROPROTECTIVE AGENT AND A RECEPTOR TYROSINE KINASE INHIBITOR ALCON, INC. (CH) 2008-07-03 WO claimed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN claimed
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN disclosed
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN disclosed
CN-101827584-A Solid dispersion product of N-aryl ureido drugs ABBOTT GMBH & CO KG 2010-09-08 CN disclosed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN disclosed