SCHEMBL3393593

SCHEMBL3393593

COc1ccc(C2(c3cc(Br)cc(OCC4CC4)c3)COC(N)=N2)cc1C.N#Cc1cc(Br)cc(OCC2CC2)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.35
KCNH2 Q12809 2/20 0.35
CTSD P07339 5/20 0.35
BACE2 Q9Y5Z0 2/20 0.34
PDE4A P27815 4/20 0.33
PDE4D Q08499 4/20 0.33
PDE4B Q07343 3/20 0.32
PDE4C Q08493 3/20 0.32
ABL1 P00519 1/20 0.30
SRC P12931 1/20 0.30
ABL2 P42684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2284332 0.93 BACE1 (0.39) BACE1KCNH2CTSDBACE2PDE4A
SCHEMBL2284328 0.93 BACE1 (0.39) BACE1KCNH2CTSDBACE2PDE4A
SCHEMBL3391476 0.88 BACE1 (0.37) BACE1KCNH2CTSDBACE2
SCHEMBL13825376 0.83 BACE1 (0.41) BACE1KCNH2CTSDBACE2PDE4A
SCHEMBL2285394 0.83 BACE1 (0.41) BACE1CTSD
SCHEMBL2285384 0.83 BACE1 (0.41) BACE1CTSD
SCHEMBL2277206 0.80 BACE1 (0.40) BACE1KCNH2CTSD
SCHEMBL2277203 0.80 BACE1 (0.40) BACE1KCNH2CTSD
SCHEMBL2283083 0.80 BACE1 (0.38) BACE1KCNH2CTSDPDE4APDE4D
SCHEMBL2283087 0.80 BACE1 (0.38) BACE1KCNH2CTSDPDE4APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed