SCHEMBL3393758

SCHEMBL3393758

COc1ccc(Cn2c(Br)nc3c(Cl)nc(N)nc32)c([N+](=O)[O-])c1OC

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 17/20 0.46
HSP90AB1 P08238 15/20 0.46
HSP90B1 P14625 4/20 0.42
TRAP1 Q12931 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3396024 0.81 HSP90AA1 (0.46) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL3395967 0.78 HSP90AA1 (0.66) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL3397111 0.76 HSP90AA1 (0.59) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1882600 0.67 TDP1 (0.47)
SCHEMBL5964706 0.67 TDP1 (0.44)
SCHEMBL11748681 0.67 KDM4E (0.44)
SCHEMBL215343 0.67 TDP1 (0.46)
SCHEMBL3394665 0.66 HSP90AB1 (0.78) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL18138425 0.66 TDP1 (0.45)
SCHEMBL14494983 0.65 POLB (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2145888-A1 Deazapurine derivatives as HSP90-Inhibitors Conforma Therapeutics Corporation (US) 2010-01-20 EP disclosed