SCHEMBL3395238

SCHEMBL3395238

CNC(=O)c1c(-c2ccc(Oc3ccc(F)cc3)cc2)oc2cc(N(CC(C)N)S(C)(=O)=O)c(C3CC3)cc12

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.64
CYP3A4 P08684 4/20 0.64
CYP2C19 P33261 4/20 0.64
KCNH2 Q12809 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395916 0.93 CYP2C9 (0.65) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL3399387 0.93 CYP2C9 (0.62) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL3393793 0.91 CYP2C9 (0.62) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL16509684 0.91 CYP2C9 (0.64) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL4093585 0.90 CYP2C9 (0.68) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL3392763 0.90 CYP2C9 (0.68) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL3399251 0.90 CYP2C9 (0.65) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL16509762 0.89 CYP2C9 (0.62) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL3396124 0.89 CYP2C9 (0.66) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL13726040 0.89 CYP2C9 (0.66) CYP2C9CYP3A4CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245023-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2010-11-03 EP claimed
WO-2009101022-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2009-08-20 WO claimed