SCHEMBL3397384

SCHEMBL3397384

COc1ccc2oc(C(Nc3ccccc3C(=O)NCCC(=O)O)C3CCCCC3)c(C#N)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
MTNR1A P48039 3/20 0.37
MTNR1B P49286 3/20 0.37
EGLN2 Q96KS0 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
ACHE P22303 3/20 0.37
BCHE P06276 2/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
POLB P06746 2/20 0.37
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
ALOX5 P09917 1/20 0.36
MAOB P27338 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL720121 0.87 GCG (0.42) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL718505 0.80 NPC1 (0.42) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL717861 0.80 NPC1 (0.39) NPC1RAB9AALDH1A1MTNR1AMTNR1B
SCHEMBL3402110 0.79 CNR1 (0.39) NPC1RAB9AKMT2APTGS1PTGS2
SCHEMBL718588 0.78 MEN1 (0.43) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL718278 0.77 NPC1 (0.43) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL720117 0.77 KMT2A (0.38) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL721161 0.76 NPC1 (0.50) NPC1RAB9AALDH1A1POLB
SCHEMBL719515 0.75 NPC1 (0.43) NPC1RAB9AALDH1A1MTNR1AMTNR1B
SCHEMBL718887 0.73 CNR2 (0.37) NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2251326-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2010-11-17 EP disclosed