SCHEMBL3397801

SCHEMBL3397801

COc1ccc(C=Cc2cccc(O[Si](C)(C)C(C)(C)C)c2)cc1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.52
RELA Q04206 1/20 0.46
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
TUBB1 Q9H4B7 4/20 0.45
TUBB4A P04350 1/20 0.45
TUBB P07437 1/20 0.45
TUBA3C P0DPH7 1/20 0.45
TUBA1B P68363 1/20 0.45
TUBA4A P68366 1/20 0.45
TUBB4B P68371 1/20 0.45
TUBB3 Q13509 1/20 0.45
TUBB2A Q13885 1/20 0.45
TUBB8 Q3ZCM7 1/20 0.45
TUBA3E Q6PEY2 1/20 0.45
TUBA1A Q71U36 1/20 0.45
TUBA1C Q9BQE3 1/20 0.45
TUBB6 Q9BUF5 1/20 0.45
TUBB2B Q9BVA1 1/20 0.45
NFE2L2 Q16236 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14363455 0.80 CYP1A1 (0.47) RELAHSP90AA1HSP90AB1TUBB1TUBB4A
SCHEMBL6158612 0.78 HSP90AA1 (0.50) NQO2RELAHSP90AA1HSP90AB1NFE2L2
SCHEMBL23923708 0.78 HSP90AA1 (0.52) NQO2RELAHSP90AA1HSP90AB1TUBB1
SCHEMBL23923707 0.78 HSP90AA1 (0.52) NQO2RELAHSP90AA1HSP90AB1TUBB1
SCHEMBL2284577 0.75 PDE4A (0.44) HSP90AA1HSP90AB1TUBB1TUBB4ATUBB
SCHEMBL1162277 0.74 HSP90AA1 (0.49) NQO2RELAHSP90AA1HSP90AB1NFE2L2
SCHEMBL20573442 0.74 HSP90AA1 (0.52) RELAHSP90AA1HSP90AB1NFE2L2CYP1A1
SCHEMBL14363441 0.74 CYP1A1 (0.73) NQO2TUBB1TUBB4ATUBBTUBA3C
SCHEMBL28672446 0.74 ABCG2 (0.47) NQO2HSP90AA1HSP90AB1TUBB1TUBB4A
SCHEMBL28672448 0.74 ABCG2 (0.47) NQO2HSP90AA1HSP90AB1TUBB1TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed