SCHEMBL3399450

SCHEMBL3399450

Cc1nc(-c2ccc(Oc3ccccc3)cc2)sc1C(=O)N1CCC(N2CCCC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.55
HRH3 Q9Y5N1 5/20 0.55
OXTR P30559 1/20 0.49
LMNA P02545 1/20 0.48
L3MBTL3 Q96JM7 4/20 0.48
L3MBTL1 Q9Y468 4/20 0.48
MBTD1 Q05BQ5 1/20 0.48
HTR2C P28335 4/20 0.48
ACHE P22303 1/20 0.46
TP53BP1 Q12888 1/20 0.46
THRA P10827 2/20 0.45
THRB P10828 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399419 0.99 HRH3 (0.56) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL13309671 0.99 HRH3 (0.56) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL3405392 0.92 CNR1 (0.55) CNR1HRH3OXTRLMNAHTR2C
SCHEMBL3405391 0.90 CNR1 (0.65) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL3403003 0.90 CNR1 (0.65) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL3398959 0.89 HRH3 (0.56) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL13309807 0.89 HRH3 (0.56) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL3405591 0.88 HRH3 (0.55) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL13309675 0.88 HRH3 (0.55) CNR1HRH3OXTRLMNAL3MBTL3
SCHEMBL13309672 0.88 HRH3 (0.47) CNR1HRH3OXTRLMNAL3MBTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed