SCHEMBL3401934

SCHEMBL3401934

O=C(NC(=O)C1CCNCC1)c1ccc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SUV39H1 O43463 3/20 0.51
PRMT1 Q99873 3/20 0.51
SMYD3 Q9H7B4 2/20 0.51
ABL1 P00519 13/20 0.49
BCR P11274 13/20 0.49
TTBK1 Q5TCY1 1/20 0.45
TTBK2 Q6IQ55 1/20 0.45
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
EPHX1 P07099 1/20 0.42
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401720 0.91 SUV39H1 (0.50) SUV39H1PRMT1SMYD3ABL1BCR
SCHEMBL3396847 0.80 ABL1 (0.50) ABL1BCRTTBK1TTBK2
SCHEMBL3397381 0.80 ABL1 (0.55) ABL1BCRTTBK1TTBK2MEN1
SCHEMBL3396560 0.79 ABL1 (0.62) ABL1BCRTTBK1TTBK2KDR
SCHEMBL3397889 0.79 ABL1 (0.59) SUV39H1PRMT1ABL1BCRTTBK1
SCHEMBL3399921 0.78 ABL1 (0.60) SUV39H1PRMT1SMYD3ABL1BCR
SCHEMBL29533110 0.78 ABL1 (0.60) SUV39H1PRMT1SMYD3ABL1BCR
SCHEMBL3398408 0.77 ABL1 (0.53) ABL1BCRTTBK1TTBK2
SCHEMBL3400770 0.77 ABL1 (0.56) SUV39H1PRMT1ABL1BCRMEN1
SCHEMBL18922428 0.77 ABL1 (0.53) SUV39H1PRMT1ABL1BCRTTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222162-A2 SMALL MOLECULE MYRISTATE INHIBITORS OF BCR-ABL AND METHODS OF USE Dana Farber Cancer Institute (US) 2010-09-01 EP claimed
WO-2009073153-A2 SMALL MOLECULE MYRISTATE INHIBITORS OF BCR-ABL AND METHODS OF USE DANA FARBER CANCER INSTITUTE (US) 2009-06-11 WO claimed