SCHEMBL3405089

SCHEMBL3405089

CCN(CC)C1CCN(C(=O)c2sc(-c3cc(C)ccc3OC)nc2C)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.46
CES2 O00748 1/20 0.40
CNR1 P21554 1/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3404365 0.95 HTR2C (0.42) HTR2CCES2MEN1KMT2ANPC1
SCHEMBL3402962 0.93 HTR2C (0.46) HTR2CCES2CNR1MEN1KMT2A
SCHEMBL3405668 0.91 HTR2C (0.44) HTR2CCES2CNR1THRBALDH1A1
SCHEMBL3399938 0.91 HTR2C (0.44) HTR2CTHRATHRBLMNA
SCHEMBL3405346 0.89 HTR2C (0.43) HTR2CCES2CNR1THRATHRB
SCHEMBL3405059 0.89 HTR2C (0.56) HTR2CCES2CNR1MEN1KMT2A
SCHEMBL3401068 0.89 HTR2C (0.48) HTR2CCES2CNR1THRATHRB
SCHEMBL3401389 0.87 HTR2C (0.42) HTR2CMEN1KMT2AALDH1A1
SCHEMBL3401212 0.87 HTR2C (0.46) HTR2CCES2CNR1THRATHRB
SCHEMBL3404372 0.86 HTR2C (0.41) HTR2CTHRBMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed