SCHEMBL3407347

SCHEMBL3407347

O=C(NCC1CC1)Oc1cnc(N2CC3=C(CN(C(=O)c4ccccc4C(F)(F)F)C3)C2)s1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCD O00767 14/20 0.47
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR2B P41595 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2296286 0.87 SCD (0.58) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL3404860 0.86 SCD (0.58) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL3406866 0.85 SCD (0.52) SCD
SCHEMBL3409272 0.84 SCD (0.49) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL3402329 0.82 SCD (0.49) SCD
SCHEMBL2290176 0.81 SCD (0.57) SCD
SCHEMBL2298045 0.77 SCD (0.77) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL2295558 0.77 SCD (0.59) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL4092350 0.76 SCD (0.73) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL12194911 0.76 SCD (0.57) SCDCYP2C9CYP2C19HTR2BMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152711-B1 2 -HETEROARYL- PYRROLO [3, 4-C]PYRROLE DERIVATIVES AND THEIR USE AS SCD INHIBITORS SANOFI AVENTIS (FR) 2010-11-24 EP disclosed