SCHEMBL3407485

SCHEMBL3407485

CC(=O)Nc1nc(CCc2ccc(CNC(=O)NN(C(=O)O)C(=O)O)cc2F)cs1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 17/20 0.51
MAOB P27338 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL973663 0.91 AOC3 (0.44) AOC3MAOBSMN1; SMN2NPC1RAB9A
SCHEMBL973662 0.88 AOC3 (0.46) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL973993 0.87 AOC3 (0.47) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL971511 0.87 AOC3 (0.57) AOC3MAOBSMN1; SMN2KMT2ANPC1
Hydrochloric Acid SCHEMBL971434 0.86 AOC3 (0.56) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL973610 0.85 AOC3 (0.57) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL972949 0.84 AOC3 (0.46) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL974261 0.81 AOC3 (0.62) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL16242040 0.81 AOC3 (0.57) AOC3MAOBSMN1; SMN2KMT2ANPC1
SCHEMBL972948 0.81 AOC3 (0.48) AOC3MAOBSMN1; SMN2KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP disclosed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO disclosed