SCHEMBL3407516

SCHEMBL3407516

Cc1ccc(-c2nc(NCCCN3CCN(C)CC3)nc3sc(OC(N)=O)c(N)c23)o1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 1/20 0.35
ADORA2A P29274 4/20 0.34
ADORA1 P30542 4/20 0.34
ICAM1 P05362 1/20 0.34
SELE P16581 1/20 0.34
SRC P12931 2/20 0.34
TLR7 Q9NYK1 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
KCNH2 Q12809 1/20 0.34
CSF1R P07333 1/20 0.34
DNMT1 P26358 2/20 0.33
DRD2 P14416 1/20 0.33
FAAH O00519 1/20 0.33
BRAF P15056 2/20 0.33
PDE4A P27815 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405349 0.88 RXFP1 (0.41) ADORA2AADORA1MEN1ALDH1A1GAA
SCHEMBL1176454 0.88 MEN1 (0.46) MEN1ALDH1A1GAAMAPTHPGD
SCHEMBL3409496 0.87 BRAF (0.40) ADORA2AADORA1MEN1ALDH1A1GAA
SCHEMBL3414240 0.84 BRAF (0.37) ADORA2AADORA1MEN1ALDH1A1GAA
SCHEMBL3409389 0.84 ADORA2A (0.35) ADORA2AADORA1TLR7MEN1ALDH1A1
SCHEMBL3407433 0.81 ADORA2A (0.33) ADORA2AADORA1TLR7MEN1ALDH1A1
SCHEMBL3406840 0.81 LIMK1 (0.42) ADORA2AADORA1MEN1ALDH1A1GAA
SCHEMBL3414093 0.80 ADORA2A (0.36) ADORA2AADORA1MEN1ALDH1A1GAA
SCHEMBL3409081 0.80 ADORA2A (0.36) ADORA2AADORA1MEN1ALDH1A1GAA
SCHEMBL3410981 0.76 LIMK1 (0.42) ADORA2AADORA1MEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP claimed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO claimed
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed