SCHEMBL3411099

SCHEMBL3411099

NCCN(OC(=O)C(F)(F)F)S(=O)(=O)c1ccc(-c2ccnc3[nH]c(Cn4ccnn4)cc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 17/20 0.51
CHUK O15111 17/20 0.51
ROCK1 Q13464 3/20 0.44
AURKB Q96GD4 1/20 0.41
AURKAIP1 Q9NWT8 1/20 0.41
CCNK O75909 1/20 0.35
CDK12 Q9NYV4 1/20 0.35
NEK1 Q96PY6 1/20 0.35
CYP2C9 P11712 1/20 0.33
CIT O14578 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3417465 0.86 CHUK (0.48) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3414337 0.83 CHUK (0.57) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3416702 0.83 IKBKB (0.59) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3412816 0.83 IKBKB (0.47) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3418266 0.82 CIT (0.47) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3411445 0.82 IKBKB (0.55) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3413538 0.81 IKBKB (0.54) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3418425 0.80 CHUK (0.43) IKBKBCHUKROCK1AURKBAURKAIP1
Trifluoroacetic Acid SCHEMBL3411097 0.80 IKBKB (0.63) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3416310 0.79 CHUK (0.56) IKBKBCHUKROCK1AURKBAURKAIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069341-B1 PYRROLO[2, 3-B]PYRIDIN-4-YL-BENZENESULFONAMIDE COMPOUNDS AS IKK2 INHIBITORS GLAXO GROUP LTD (GB) 2010-12-29 EP disclosed