SCHEMBL3412461

SCHEMBL3412461

Cc1ccc(-c2ccsc2C(=O)N2C[C@@H]3C[C@@H]3[C@H]2CN)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.41
HCRTR2 O43614 5/20 0.41
BCAT2 O15382 1/20 0.33
ALDH1A1 P00352 3/20 0.32
TSHR P16473 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 1/20 0.32
S1PR1 P21453 1/20 0.32
S1PR5 Q9H228 1/20 0.32
MAPT P10636 3/20 0.32
MAPK1 P28482 2/20 0.32
HSD17B10 Q99714 1/20 0.32
EGFR P00533 1/20 0.31
TYMS P04818 1/20 0.31
LTA4H P09960 1/20 0.31
VDR P11473 1/20 0.31
SRC P12931 1/20 0.31
CTSK P43235 1/20 0.31
KDM1A O60341 2/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1340425 0.90 PTGS1 (0.38) HCRTR1HCRTR2BCAT2ALDH1A1TSHR
SCHEMBL3413488 0.88 HCRTR1 (0.43) HCRTR1HCRTR2BCAT2ALDH1A1TSHR
SCHEMBL1340215 0.83 HCRTR2 (0.33) HCRTR1HCRTR2POLBS1PR1S1PR5
SCHEMBL3412456 0.83 HCRTR1 (0.39) HCRTR1HCRTR2BCAT2ALDH1A1TSHR
SCHEMBL2803127 0.83 HCRTR1 (0.41) HCRTR1HCRTR2BCAT2ALDH1A1TSHR
SCHEMBL2927516 0.80 CYP46A1 (0.40) HCRTR1HCRTR2KDM1A
SCHEMBL3417003 0.80 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL2931897 0.80 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL2924236 0.80 KDM1A (0.35) HCRTR1HCRTR2POLBS1PR1S1PR5
SCHEMBL3417319 0.79 CA12 (0.39) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185512-B1 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-12-29 EP claimed
EP-2185512-B1 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-12-29 EP disclosed