SCHEMBL3414868

SCHEMBL3414868

O=C(Cc1cc2c(-c3ccc(S(=O)(=O)NCCOC(=O)C(F)(F)F)cc3)ccnc2[nH]1)N1CCCC1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 14/20 0.55
CHUK O15111 14/20 0.55
ROCK1 Q13464 3/20 0.55
NEK1 Q96PY6 5/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3414866 0.89 IKBKB (0.59) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3414579 0.88 IKBKB (0.65) IKBKBCHUKROCK1NEK1CYP2C9
Trifluoroacetic Acid SCHEMBL3412810 0.87 IKBKB (0.67) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3410064 0.85 IKBKB (0.75) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3607022 0.85 IKBKB (0.58) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3414009 0.82 IKBKB (0.56) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3417481 0.82 IKBKB (0.77) IKBKBCHUKROCK1NEK1CYP2C9
SCHEMBL3617126 0.81 IKBKB (0.68) IKBKBCHUKROCK1NEK1CYP2C9
Trifluoroacetic Acid SCHEMBL3415936 0.80 IKBKB (0.51) IKBKBCHUKROCK1CYP2C9
SCHEMBL3413149 0.80 IKBKB (0.73) IKBKBCHUKROCK1NEK1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069341-B1 PYRROLO[2, 3-B]PYRIDIN-4-YL-BENZENESULFONAMIDE COMPOUNDS AS IKK2 INHIBITORS GLAXO GROUP LTD (GB) 2010-12-29 EP disclosed