SCHEMBL3418471

SCHEMBL3418471

C=CC(C=O)c1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.43
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
TGM2 P21980 3/20 0.34
F13A1 P00488 1/20 0.34
LMNA P02545 1/20 0.34
TGM1 P22735 1/20 0.34
TGM3 Q08188 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
PYCR1 P32322 1/20 0.32
HTR2A P28223 1/20 0.32
ALOX5 P09917 1/20 0.32
CNR1 P21554 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1129069 0.86 CYP2A6 (0.42) CYP2C19CYP1A2CYP2A6SMN1; SMN2HTR2A
SCHEMBL27372777 0.78 HSD17B10 (0.39) CYP2A6LMNA
SCHEMBL11042692 0.78 MAPT (0.42) CYP2C19CYP1A2LMNA
SCHEMBL1335929 0.77 CYP2D6 (0.41) CYP2C19CYP2A6LMNA
SCHEMBL28583238 0.75 CYP3A4 (0.43)
SCHEMBL27373192 0.75 CYP2C19 (0.42) CYP2C19CYP1A2CYP2A6TGM2F13A1
SCHEMBL12333611 0.74 SLC6A2 (0.37) CYP2C19LMNASMN1; SMN2
SCHEMBL321965 0.70 CYP2A6 (0.40) CYP2C19CYP1A2CYP2A6SMN1; SMN2HTR2A
SCHEMBL22590138 0.70 CYP2A6 (0.40) CYP2C19CYP1A2CYP2A6SMN1; SMN2HTR2A
SCHEMBL7131926 0.70 CYP2C19 (0.42) CYP2C19CYP1A2CYP2A6TGM2F13A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1468994-B1 Process for preparing cyclic amine substituted phenyl-alkyl-ketones BASF SE (DE) 2010-11-24 EP disclosed
EP-0805152-B1 Cyclic amine substituted phenyl-alkyl-ketone and process for its preparation CIBA SC HOLDING AG (CH) 2005-06-08 EP disclosed
EP-1468994-A1 Process for preparing cyclic amine substituted phenyl-alkyl-ketones Ciba SC Holding AG (CH) 2004-10-20 EP disclosed
US-6191182-B1 SUBJECTING P-HALOPHENYL ALKYL KETONE TO AMINOLYSIS WITH CYCLIC SECONDARY AMINE TO FORM CYCLIC AMINE-SUBSTITUTED PHENYL ALKYL KETONE; HALOGINATION AND REACTING WITH AMINE COMPOUND; STEVENS REARRANGEMENT UNDER BASIC CONDITION CIBA SPECIALTY CHEMCIALS CORPORATION 2001-02-20 US disclosed
US-5977357-A Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof CIBA SPECIALTY CHEMICAL CORPORATION (US) 1999-11-02 US disclosed
US-5795985-A Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-08-18 US disclosed
EP-0805152-A2 Cyclic amine substituted phenyl-alkyl-ketone and process for its preparation Ciba SC Holding AG (CH) 1997-11-05 EP disclosed