SCHEMBL3425262

SCHEMBL3425262

Cc1cc(NC(=O)C(C)(C)NC(=O)c2ccc(Cl)s2)ccc1C(=O)N1CCCN(C)CC1

nearest known ligand 0.86

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.86
AR P10275 3/20 0.53
KMT2A Q03164 5/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
EPHX2 P34913 1/20 0.38
PDE7A Q13946 1/20 0.38
CNR2 P34972 1/20 0.37
NPY2R P49146 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3423791 0.96 F10 (0.86) F10ARKMT2ALMNAMAPK1
SCHEMBL3427505 0.93 F10 (1.00) F10ARKMT2ALMNAMAPK1
SCHEMBL3426052 0.92 F10 (0.98) F10ARKMT2AALDH1A1HPGD
SCHEMBL3425291 0.92 F10 (0.98) F10ARKMT2AALDH1A1HPGD
SCHEMBL3427677 0.90 F10 (0.69) F10ARKMT2ALMNAHPGD
SCHEMBL3427996 0.89 F10 (0.86) F10ARKMT2AALDH1A1HPGD
SCHEMBL3424566 0.89 F10 (0.86) F10ARKMT2AALDH1A1HPGD
SCHEMBL3426538 0.88 F10 (0.86) F10ARKMT2ALMNAMAPK1
SCHEMBL3424771 0.87 F10 (0.82) F10ARKMT2ALMNAMAPK1
SCHEMBL3426142 0.87 F10 (0.84) F10ARKMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732466-B2 Substituted thiophene carboxamides, process for their preparation and their use as medicaments BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-08 US disclosed
US-7732466-B2 Substituted thiophene carboxamides, process for their preparation and their use as medicaments BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-08 US disclosed
US-7732466-B2 Substituted thiophene carboxamides, process for their preparation and their use as medicaments BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-08 US disclosed
US-20060293300-A1 New substituted thiophene carboxamides, process for their preparation and their use as medicaments BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-12-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060293300-A1 New substituted thiophene carboxamides, process for their preparation and their use as medicaments OTC, TPMT, ABCG2 F10 1901/4885AR 3491/4885KMT2A 2674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.