SCHEMBL3427558

SCHEMBL3427558

CN1CCCC1Cn1cc(C(=O)N2CCC3(CC2)OCc2ccncc23)c2ccc(Cl)cc21

nearest known ligand 0.81

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 12/20 0.81
CNR1 P21554 3/20 0.45
OXTR P30559 1/20 0.43
CNR2 P34972 1/20 0.39
IL1B P01584 1/20 0.39
P2RX7 Q99572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2512004 1.00 AVPR1A (0.81) AVPR1ACNR1OXTRCNR2IL1B
SCHEMBL2524189 0.91 AVPR1A (0.68) AVPR1ACNR1OXTRCNR2
SCHEMBL2524187 0.91 AVPR1A (0.68) AVPR1ACNR1OXTRCNR2
SCHEMBL4361697 0.90 AVPR1A (1.00) AVPR1ACNR1OXTRCNR2
SCHEMBL4357753 0.90 AVPR1A (1.00) AVPR1ACNR1OXTRCNR2
SCHEMBL2515628 0.88 AVPR1A (0.64) AVPR1ACNR1OXTRCNR2IL1B
SCHEMBL3393027 0.86 AVPR1A (0.81) AVPR1ACNR1OXTRCNR2IL1B
Hydrochloric Acid SCHEMBL2515633 0.85 AVPR1A (0.80) AVPR1ACNR1OXTRCNR2IL1B
SCHEMBL2514280 0.85 AVPR1A (0.79) AVPR1ACNR1OXTRCNR2IL1B
SCHEMBL2519890 0.85 AVPR1A (0.79) AVPR1ACNR1OXTRCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125827-B1 AZASPIRO DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-11-03 EP claimed