SCHEMBL3428634

SCHEMBL3428634

CCc1nc2c(cnn2CC)c(NC2CCOCC2)c1CNC(=O)NCc1ccc(F)c(-c2cccc(CN3CCN(C(=O)O)[C@@H](C)C3)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.43
CHRM3 P20309 16/20 0.43
CHRM2 P08172 6/20 0.39
CHRM1 P11229 6/20 0.39
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350728 0.96 PDE4B (0.42) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4190920 0.95 CHRM3 (0.49) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4098861 0.95 PDE4B (0.44) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4346720 0.94 PDE4B (0.41) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4106585 0.94 CHRM3 (0.46) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4355753 0.94 PDE4B (0.41) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4190753 0.94 PDE4B (0.48) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL3430634 0.93 CHRM3 (0.45) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL3425551 0.92 PDE4B (0.42) PDE4BCHRM3
SCHEMBL4349671 0.92 PDE4B (0.40) PDE4BCHRM3CHRM2CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2249830-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS Glaxo Group Limited (GB) 2010-11-17 EP disclosed
WO-2009100170-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed