SCHEMBL3430901

SCHEMBL3430901

N#Cc1cc(-c2nc(-c3ccc4c(c3)CCN(C(=O)CNC(=O)O)CC4)no2)ccc1OC(CF)CF

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.61
S1PR3 Q99500 7/20 0.61
KCNH2 Q12809 2/20 0.56
S1PR5 Q9H228 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3431138 0.91 S1PR1 (0.74) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2125106 0.90 S1PR1 (0.56) S1PR1S1PR3KCNH2
SCHEMBL2122394 0.89 S1PR1 (0.62) S1PR1S1PR3KCNH2S1PR5
SCHEMBL3430660 0.87 S1PR1 (0.55) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2122681 0.85 S1PR1 (0.60) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2128935 0.85 S1PR1 (0.59) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2130295 0.84 S1PR1 (0.61) S1PR1S1PR3KCNH2S1PR5
SCHEMBL3430908 0.82 S1PR1 (0.55) S1PR1S1PR3KCNH2
SCHEMBL2605649 0.82 S1PR1 (0.67) S1PR1S1PR3KCNH2
SCHEMBL3430836 0.81 S1PR1 (0.70) S1PR1S1PR3KCNH2S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed