Warfarin

Warfarin

SCHEMBL34347

CC(=O)CC(c1ccccc1)c1c(O)c2ccccc2oc1=O.[NaH]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

VKORC1

The experimentally established mechanism targets of Warfarin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VKORC1 known ✓ Q9BQB6 3/20 0.97
CYP2C9 P11712 10/20 0.97
ALB P02768 2/20 0.97
HSD17B10 Q99714 2/20 0.97
KDM4E B2RXH2 1/20 0.97
ALDH1A1 P00352 1/20 0.97
PCSK7 Q16549 1/20 0.97
MEN1 O00255 1/20 0.97
KMT2A Q03164 1/20 0.97
NR1I2 O75469 1/20 0.75
NR3C1 P04150 1/20 0.75
ADRA1A P35348 1/20 0.75
KCNH2 Q12809 1/20 0.75
CYP3A4 P08684 1/20 0.73
BRD4 O60885 1/20 0.67
NQO1 P15559 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Warfarin SCHEMBL28534047 1.00 CYP2C9 (0.97) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL5483689 1.00 CYP2C9 (0.97) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL8332637 1.00 CYP2C9 (0.97) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL13278154 1.00 CYP2C9 (0.97) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL29400364 0.99 CYP2C9 (1.00) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL3689 0.99 CYP2C9 (1.00) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL662875 0.99 CYP2C9 (1.00) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL4439794 0.99 CYP2C9 (1.00) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL2139452 0.99 CYP2C9 (1.00) CYP2C9VKORC1ALBHSD17B10KDM4E
Warfarin SCHEMBL3792087 0.99 CYP2C9 (1.00) CYP2C9VKORC1ALBHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6738 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026087732-A1 LIQUID, MULTI-DOSE, READY-TO-USE WARFARIN COMPOSITION AND USE HYLORIS DEVELOPMENTS SA (BE) 2026-04-30 WO claimed
EP-4688415-A1 DOUBLE LAYER TUBING FOR IV INFUSION SETS CareFusion 303, Inc. (US) 2026-02-11 EP claimed
CN-120005821-A Immune cell culture method 上海华颜医药科技有限公司 2025-05-16 CN claimed
WO-2025022245-A1 A READY-TO-USE ORAL LIQUID FORMULATION OF WARFARIN SODIUM LIQMEDS WORLDWIDE LIMITED (GB) 2025-01-30 WO claimed
US-20240374769-A1 LIGHT ACTIVATED CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY 2024-11-14 US claimed
WO-2024233595-A1 LIGHT ACTIVATED CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY (US) 2024-11-14 WO claimed
CN-118924473-A Gingival bleeding animal model, method and application of chronic periodontitis with coagulation disorder 上海交通大学医学院附属第九人民医院 2024-11-12 CN claimed
CN-118834562-A Poria cocos acidic polysaccharide chiral stationary phase and application thereof 云南中医药大学 2024-10-25 CN claimed
US-20240325623-A1 DOUBLE LAYER TUBING FOR IV INFUSION SETS CAREFUSION 303, INC. 2024-10-03 US claimed
WO-2024205867-A1 DOUBLE LAYER TUBING FOR IV INFUSION SETS CAREFUSION 303, INC. (US) 2024-10-03 WO claimed
WO-2001028555-A1 EMULSION COMPOSITIONS FOR POLYFUNCTIONAL ACTIVE INGREDIENTS LIPOCINE, INC. (US) 2001-04-26 WO claimed
EP-1089992-A1 SYNTHESES BASED ON 2-HYDROXYACETOPHENONE Hoechst Celanese Corporation (US) 2001-04-11 EP claimed
EP-1089992-A4 SYNTHESES BASED ON 2-HYDROXYACETOPHENONE HOECHST CELANESE CORP (US) 2001-04-11 EP claimed
WO-2001012155-A1 COMPOSITIONS AND METHODS FOR ENHANCED ABSORPTION OF HYDROPHILIC THERAPEUTIC AGENTS LIPOCINE, INC. (US) 2001-02-22 WO claimed
WO-2000024386-A1 METHOD OF MAKING PRESSURE SENSITIVE ADHESIVE MATRIX PATCHES CONTAINING HYDROPHILIC SALTS OF DRUGS THERATECH, INC. (US) 2000-05-04 WO claimed
US-5935802-A Method of assaying a blood sample for prothrombin EVANSTON NORTHWESTERN HEALTHCARE RESEARCH INSTITUTE (US) 1999-08-10 US claimed
CN-1194781-A Method for obtainment of biological rodenticide BIOLOG FARMACEUTICOS LABIOFAM (CU) 1998-10-07 CN claimed
US-5696274-A Syntheses based on 2-hydroxyacetophenone HOECHST CELANESE CORPORATION (US) 1997-12-09 US claimed
WO-1997024347-A1 SYNTHESES BASED ON 2-HYDROXYACETOPHENONE HOECHST CORPORATION (US) 1997-07-10 WO claimed
US-5328453-A Method for enhancing transdermal drug delivery of electrical drug applicators DRUG DELIVERY SYSTEMS INC. (US) 1994-07-12 US claimed