SCHEMBL3435205

SCHEMBL3435205

COC(=O)c1cccc2cn(C3CCCN(C(=O)OCc4ccccc4)C3)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
JAK2 O60674 3/20 0.42
JAK1 P23458 3/20 0.42
TYK2 P29597 2/20 0.42
JAK3 P52333 2/20 0.42
HTT P42858 1/20 0.42
LCK P06239 2/20 0.41
PDE4B Q07343 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
BCL9 O00512 2/20 0.41
CTNNB1 P35222 2/20 0.41
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204967 0.75 LCK (0.46) SMN1; SMN2NPC1RAB9AJAK2JAK1
SCHEMBL29138124 0.73 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9AJAK2JAK1
SCHEMBL206309 0.73 HSD17B10 (0.55) SMN1; SMN2NPC1RAB9AHTTHSD11B1
SCHEMBL1441223 0.72 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AJAK2JAK1
SCHEMBL20129713 0.72 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AJAK2JAK1
SCHEMBL3678408 0.71 TMEM97 (0.57) SMN1; SMN2NPC1RAB9ACYP2C19TMEM97
SCHEMBL11916703 0.71 PDE4B (0.57) SMN1; SMN2NPC1RAB9AJAK2JAK1
SCHEMBL22765331 0.71 TMEM97 (0.57) SMN1; SMN2NPC1RAB9ACYP2C19TMEM97
SCHEMBL27678403 0.71 PDE4B (0.57) SMN1; SMN2NPC1RAB9AJAK2JAK1
SCHEMBL4982385 0.71 PDE4B (0.55) SMN1; SMN2NPC1RAB9AJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed